Trametinib are cas 871700-17-3

Trametinib are cas 871700-17-3
Khoom Taw qhia:
Catalog Tsis yog.: SS122599
CAS TSIS MUAJ .: 871700-17-3
Purity (HPLC): 99% min
Khoom npe: trametinib
Molecular Cov Qauv: C26h23Fin5O4
Molecular hnyav: 615.39
Xa kev nug
Kev tsis
Hauj lwm lawm

 

Cov lus qhia

 

Kev tshwm sim Tawm - hmoov dawb
Purity (hplc) 99% min
1h nmr Sib xws rau cov qauv

 

Cov Ntaub Ntawv Thauj

 

Chaw ua uas tsis tau haus

Kev qhia tshwj xeeb

UN NUM

 

Hom

 

Cov Pab Pawg

 

Hs code

2933599099304

Ruaj khov & rov ua

Cov khoom lag luam ruaj khov nyob rau hauv cov qauv ambient ambient.

Chaw ntim khoom

-20 degC

Mob kom tsis txhob

 

Lub thawv

 

 

Cov ntaub ntawv raug

 

Chaw ua uas tsis tau haus

Kev qhia tshwj xeeb

Lub peev xwm

 

Hov ntau

 

Lub teb chaws tseem ceeb

 

Peev Xwm / Batch

 

Paub lawm

Ntau lawm txij xyoo 2015

Ntxiv rau

 

 

 

 

Cov Ntawv Thov

 

Trametinib feem ntau siv los ua cov tshuaj tiv thaiv anticancer, tshwj xeeb xws li ib tug mek inhibitor nyob rau hauv kev kho ntawm melanoma thiab lwmyam cancer nrog rau kev sib tsoo. Nws yog muab ua ke ua ib feem ntawm kev kho ua ke los yog ua kev kho mob monotherapy rau inhibit qog cell proliferation. Tsis tas li ntawd, trametinib yog siv nyob rau hauv preclinical thiab kev tshawb nrhiav hauv kev soj ntsuam mus kawm cov txheej txheem transduction barduction, thiab cov tshuaj tiv thaiv, thiab cov tshuaj tiv thaiv nyob rau hauv oncology.

 

Cov txiaj ntsig

 

Trametinib muab cov kev xaiv heev nyob rau hauv Mek1 thiab Mek2 Enzymes, muaj txiaj ntsig zoo rau Mapk / ERK signing txoj kev, uas feem ntau tsis sib thooj hauv qee lub qog. Cov tshuab ntsuas no tso cai rau txo cov qog kom txo qis ntawm - phiaj cuam tshuam piv rau cov kws khomob kho kom zoo nkauj. Nws qhov rooj ntawm qhov ncauj thiab kev ua tau zoo rau kev kho mob txhim kho cov txiaj ntsig kho tau thiab muab ib qho kev xaiv muaj txiaj ntsig zoo rau cov neeg mob uas muaj tshwj xeeb caj ces.

 

Tag

 

Trametinib yog qhov tseem ceeb tshaj plaws kev kho mob hauv oncology, muab xaiv mess incology, muab kev xaiv Mexis incibition rau kev kho mob cancers ntawm braf mutations. Nws qhov tshwj xeeb, cov txiaj ntsig, thiab cov kws kho mob tseem ceeb rau kev tshawb fawb thiab kev tshawb fawb txuas ntxiv hauv cov tswv yim anticancer niaj hnub no.

 

 

Cim npe nrov: Trametinib are Cas 871700-17-3, Tuam Tshoj Trametinib are Cas 871700-17-3 Cov Chaw Tsim Tshuaj, Chaw Tsim Tshuaj, Hoobkas

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