Cov lus qhia
| Kev tshwm sim | Tawm - hmoov dawb |
| Purity (hplc) | 99% min |
| 1h nmr | Sib xws rau cov qauv |
Cov Ntaub Ntawv Thauj
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Chaw ua uas tsis tau haus |
Kev qhia tshwj xeeb |
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UN NUM |
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Hom |
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Cov Pab Pawg |
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Hs code |
2933599099304 |
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Ruaj khov & rov ua |
Cov khoom lag luam ruaj khov nyob rau hauv cov qauv ambient ambient. |
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Chaw ntim khoom |
-20 degC |
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Mob kom tsis txhob |
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Lub thawv |
Cov ntaub ntawv raug
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Chaw ua uas tsis tau haus |
Kev qhia tshwj xeeb |
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Lub peev xwm |
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Hov ntau |
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Lub teb chaws tseem ceeb |
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Peev Xwm / Batch |
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Paub lawm |
Ntau lawm txij xyoo 2015 |
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Ntxiv rau |
Cov Ntawv Thov
Trametinib feem ntau siv los ua cov tshuaj tiv thaiv anticancer, tshwj xeeb xws li ib tug mek inhibitor nyob rau hauv kev kho ntawm melanoma thiab lwmyam cancer nrog rau kev sib tsoo. Nws yog muab ua ke ua ib feem ntawm kev kho ua ke los yog ua kev kho mob monotherapy rau inhibit qog cell proliferation. Tsis tas li ntawd, trametinib yog siv nyob rau hauv preclinical thiab kev tshawb nrhiav hauv kev soj ntsuam mus kawm cov txheej txheem transduction barduction, thiab cov tshuaj tiv thaiv, thiab cov tshuaj tiv thaiv nyob rau hauv oncology.
Cov txiaj ntsig
Trametinib muab cov kev xaiv heev nyob rau hauv Mek1 thiab Mek2 Enzymes, muaj txiaj ntsig zoo rau Mapk / ERK signing txoj kev, uas feem ntau tsis sib thooj hauv qee lub qog. Cov tshuab ntsuas no tso cai rau txo cov qog kom txo qis ntawm - phiaj cuam tshuam piv rau cov kws khomob kho kom zoo nkauj. Nws qhov rooj ntawm qhov ncauj thiab kev ua tau zoo rau kev kho mob txhim kho cov txiaj ntsig kho tau thiab muab ib qho kev xaiv muaj txiaj ntsig zoo rau cov neeg mob uas muaj tshwj xeeb caj ces.
Tag
Trametinib yog qhov tseem ceeb tshaj plaws kev kho mob hauv oncology, muab xaiv mess incology, muab kev xaiv Mexis incibition rau kev kho mob cancers ntawm braf mutations. Nws qhov tshwj xeeb, cov txiaj ntsig, thiab cov kws kho mob tseem ceeb rau kev tshawb fawb thiab kev tshawb fawb txuas ntxiv hauv cov tswv yim anticancer niaj hnub no.
Cim npe nrov: Trametinib are Cas 871700-17-3, Tuam Tshoj Trametinib are Cas 871700-17-3 Cov Chaw Tsim Tshuaj, Chaw Tsim Tshuaj, Hoobkas

