Cov lus qhia tshwj xeeb ntawm Tadalafil 丨 CAS 171596-29-5
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Ntiag tug |
Kev qhia tshwj xeeb |
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Teem nqi |
EP11. 0 |
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Kev tshwm sim |
Dawb lossis yuav luag dawb hmoov |
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Lam xav |
97.5% thiab 102.5%, xam ntawm cov dej qhuav |
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So |
Dawb soluble nyob rau hauv duethyl sulfoxide, me ntsis soluble hauv dichloromshane, kev ua insoluble hauv dej |
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TSHWJ XEEB REGICCER |
78. {{{0 degree - 84. {{}}} Degree |
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HPLC |
Lub sijhawm khaws cia ntawm qhov kev daws teeb meem loj ntawm cov qauv daws teeb meem, raws li tau txais hauv kev sim rau enantiomeric thiab diastereomeric purity |
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Organic Impurities |
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Tus kheej impurities |
0. 1% Max |
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Tag nrho cov impurities |
0. 3% Max |
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Tus pab mov |
|
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6R, 12AS diastereomer |
0. 1% Max |
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6s, 12as enantiomer |
0. 1% Max |
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6s, 12ar diastereomer |
0. 1% Max |
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Residual cov kuab tshuaj |
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Mellylamine |
{{0 {}}. 163% Max |
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Methanol |
0. 3% Max |
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Acetonitrile |
{{0 {}}. 041% Max |
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IsoPropanol |
{{0 {}}. 5% Max |
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Ethyl Acetate |
{{0 {}}. 5% Max |
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Dmf |
0. 088% Max |
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Residue ntawm ignition |
0. 1% Max |
|
Poob rau ziab |
{{0 {}}. 5% Max |
Tadalafil 丨 CAS 171596-29-5}}}}}}}}}) Inhibital siv feem ntau rau kev kho mob erectile (ed) thiab benign prostatic hyperplasia (bpph). Tadalafil ua haujlwm los ntawm inhibiting PDE5 enzyme, uas tswj cov ntshav hauv cov nqaij mos thiab prostate, yog li kev txhim kho cov tsos mob ntawm ed thiab bph. Nws tau pom zoo tau pom zoo los ntawm Asmeskas FDA xyoo 2003 thiab muaj txij li los ua cov tshuaj siv rau erectile kawg.
Cov ntawv thov ntawm Tadalafil 丨 CAS 171596-29-5
1. Erectile kawg (ed)
● Ciais feem ntau siv los kho erectile kawg (ED), ib qho xwm txheej uas tus txiv neej tsis tuaj yeem ua tiav lossis tswj hwm qhov erection txaus rau kev sib deev.
● Nws ua haujlwm los ntawm kev nce ntshav ntws mus rau qhov chaw mos los ntawm kev cuam tshuam txog kev cuam tshuam ntawm PDE5, cov protein uas tswj cov ntshav los ntawm tawg guanosine monophosphate (CGMP). Qhov no tso cai rau lub caij nyoog ntev thiab erection hauv kev teb rau kev sib deev.
● Ntev ntev ntawm kev nqis tes ua: ib qho ntawm cov txiaj ntsig tseem ceeb ntawm lwm tus PDE5 Inhibitors (uas yog nws lub neej ntev ntawm kwv yees li 17.5 teev, cia rau kev cuam tshuam uas muaj peev xwm kav ntev txog 36 teev. Qhov no tso cai rau ntau qhov sib deev sib deev.
2. Benign prostatic hyperplasia (bpph)
● Tadalafil tseem siv los kho benign prostatic hyperplasia (BPP), ib qho xwm txheej ntawm tus mob prostsate, uas tuaj yeem ua rau etrinary nyuaj, xws li nquag tso zis, kev kub ntxhov, thiab cov zis tsis muaj zog, thiab cov zis tsis muaj zog
Los ntawm kev cuam tshuam PDE5, cialis relaxing cov leeg du hauv prostate thiab zais zis, uas pab txo cov tsos mob BPH thiab txhim kho kev nyab xeeb.
3. Pulmonary Arterial Tawg (PAH)
● Tadalafil raug pom zoo rau kev kho mob ntawm bulmonary bypection (PAH), tus mob uas muaj ntshav siab nyob rau hauv lub ntsws 'arteries.
It Nws ua haujlwm los ntawm cov hlab ntshav kom txaus, thiab kev ua haujlwm ntawm lub peev xwm ntawm cov neeg mob nrog PAH.
● Ciais feem ntau tau muab rau hauv qab lub npe sib txawv rau pah kho (Adcirca).
4. Cov ntawv sau npe tawm
● Raynud tus kab mob: Cialis tau tshawb nrhiav rau kev siv hauv kev kho cov kab mob sib txawv, uas cov hlab ntshav hauv qhov kawg tsis muaj mob rau kev teb txias lossis ntxhov siab.
Ensogathabete Neuropathy: Qee cov kev tshawb fawb qhia tau tias Tadalafil tuaj yeem muaj lub luag haujlwm muaj peev xwm tswj hwm ntshav qab zib Neuropathy, txawm hais tias qhov no tseem tab tom tshawb nrhiav.
Cov txiaj ntsig ntawm tadalafil 丨 CAS 171596-29-5
1. Kev kho mob rau Ed
● Ciais yog paub rau nws txoj kev ua nrawm nrawm ntawm 30 feeb), thiab nws lub sijhawm ntev ntawm cov sij hawm, muab lub qhov rais ntawm lub sijhawm ntev txog 36 teev ntawm cov hauj lwm zoo.
● Cov tshuaj kho mob uas tsis zoo li lwm yam erectile tsis tau yuav tsum tau ua kom tiav sijhawm ua ntej kev sib deev, ua rau nws yooj yim rau kev siv kev sib deev.
2. Txhim Kho Lub Neej Zoo
Tshaj tawm cov txiaj ntsig ntawm lub cev, Tadalafil tau pom tias txhim kho kev ntseeg hlwb los ntawm kev txhim kho kev ntseeg siab thiab txo kev ntxhov siab cuam tshuam nrog kev ua tau zoo.
● Los ntawm kev kho bph, nws txhim kho lub neej zoo hauv txiv neej kev txom nyem los ntawm kev tso zis qis dua (Luts), ua kom muaj kev cuam tshuam zoo dua thiab cuam tshuam tsawg dua rau cov dej num txhua hnub.
3. Dual kev txiav txim rau ed thiab bph
Muaj peev xwm los kho ob qho kev ua tsis tau erectile thiab benign prostatic hyperplasia hauv ib qho tshuaj yog qhov txiaj ntsig tseem ceeb rau cov txiv neej uas raug mob los ntawm ob qho tib si.
● Tadalafil tuaj yeem pab cov txiv neej tswj kev noj qab haus huv thiab cov tso zis, uas ua rau txhim kho tag nrho kev noj qab haus huv thiab kev nplij siab.
4. Kev Nyab Xeeb Kev Nyab Xeeb
● Tadalafer 丨 CAS 171596-29-5 yog feem ntau yog qhov zoo ntawm sab mob me me piv tau piv rau lwm yam tshuaj rau erectile kawg.
Lub neej ntev ib nrab-lub neej yuav tsum tau noj tshuaj tsawg dua, thiab cov kev xaiv tshuaj txhua hnub pub rau cov txiv neej nrog cov tsos mob lossis bph.
Tag
Tadalafil 丨 CAS 171596-29-5 Cov tshuaj zoo rau kev kho mob erectile rau kev kho erectile siab, thiab pulmonary arterial ntshav siab. Nws lub sijhawm ntev ntawm kev nqis tes ua (txog li 36 teev) ua rau nws yooj yim dua piv rau lwm cov tshuaj erectile tsis sib xws. Nws muaj qhov txiaj ntsig ntxiv ntawm kev kho ob qho kev sib daj sib deev thiab tso zis rau cov txiv neej muaj bph, txhim kho kev ua kom zoo ntawm lub neej. Thaum feem ntau muaj kev nyab xeeb, nws yuav tsum tau siv nyob rau hauv kev saib xyuas kev saib xyuas, tshwj xeeb yog nyob rau hauv cov tib neeg uas muaj qee yam mob.
Cim npe nrov: Tadalafil 丨 cas 171596-29-5}}, Tuam Tshoj Tadalafil 丨 CAS 171596-29-5 Cov chaw tsim khoom, cov chaw tsim khoom, Hoobkas

