Cov lus qhia tshwj xeeb ntawm Sumatriptan succminate 丨 103628-48-4
|
Qib: |
EP9. {0 |
|
Zog: |
Dawb lossis yuav luag dawb hmoov |
|
Assay: |
97.5% - 102% (cov khoom siv anhydrot) |
|
Solubility: |
Dawb soluble hauv dej, sparingly soluble hauv methanol, tau ua insoluble hauv methylene chloride |
|
Daim qhia npe: |
IR: Yuam kom sumatriptan succinate CLS |
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Ph: |
4.5 – 5.3 |
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Absorbance: |
0. 1 Max |
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Impurity a: |
{{0 {}}. 6% Max |
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Impurity h: |
0. 3% Max |
|
Impurity b, c, D: |
Txhua 0. 5% Max |
|
Ipurity E: |
0. 15% Max |
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Unspecified impurities: |
0. 1% Max |
|
Tag nrho cov impurity: |
{{0 {}}. 6% Max |
|
Dej: |
1. {0 max |
|
Sulphated tshauv: |
0. 1% Max |
|
Residual cov kuab tshuaj: |
Methanol: 0. 3% Max |
Sumatriptan succinate 丨 cas 103628-48-4 yog lub succinate ntsev ({} hteptor agonist feem ntau siv nyob rau hauv kev kho mob migraine thiab cluster taub hau. Nws yog pob kws nyob hauv chav kawm ntawm Triptans, yeeb siv tshuaj tshwj xeeb los tsom cov pathophysiology ntawm migraines.
Cov ntawv thov tseem ceeb ntawm Sumatriptan succuate 丨 cas 103628-48-4
1. Migraine Kev Kho Mob
Sumatriptan succinate 丨 cas 103628-48-4} feem ntau tau muab tshuaj rau kev kho mob hnyav Nws ua haujlwm los ntawm kev txhawb nqa serotonin cov receptors nyob rau hauv lub hlwb, uas ua nyob rau hauv vasoconstratic ntawm dhuav cov ntshav hlab ntsha-ib qho ntawm cov ua rau mob plab.
2. Cluster Headache nyem
Ntxiv rau migraines, nws kuj tseem siv rau kev kho mob hnyav ntawm pawg tiv thaiv cluster, ib hom mob taub hau heev uas tshwm sim hauv cov qauv kev nyiam ua neeg.
3. Tshuaj Kho Mob
Muaj nyob rau hauv ntau cov kev siv tshuaj suav nrog:
● Cov ntsiav tshuaj ntawm qhov ncauj
● Subcutaneys txhaj
● Nasal tshuaj tsuag
● Transdermal patches
Txhua txoj kev yog txiav kom muaj kev cuam tshuam sai sai ntawm kev nqis tes ua raws li qhov hnyav thiab sijhawm ntawm cov tsos mob migraine.
4. Tshawb nrhiav thiab kev txhim kho
Sumatriptan succmined tseem muaj dav siv nyob rau hauv chaw soj ntsuam cov kev tshawb fawb rau:
● Nkag siab txog kev siv tshuab
Tsim cov khoom siv tshiab
● Sib piv ua tau zoo nrog cov triptans tshiab lossis kev kho mob
Cov txiaj ntsig ntawm SumatRiptan succminate 丨 cas 103628-48-4
✅ Kev Pab Dawb Ceev Ceev
Nws feem ntau pib daws cov tsos mob hauv 30 mus rau 60 feeb, tshwj xeeb tshaj yog nyob rau hauv cov ntawv txhaj lossis intranasal.
✅ Lub Hom Phiaj
Tsis zoo li cov kev mob mob rau kev mob siab rau kev ua txhaum cai lij choj serotonin receptors cuam tshuam hauv cov migraines, ua rau nws muaj txiaj ntsig zoo.
Of Cov kev xaiv ntau ntau
Qhov muaj ntawm ntau txoj kev tswj hwm tso cai rau cov tib neeg raws li cov tsos mob pib ntawm kev ceev thiab tus neeg mob nyiam.
✅ Cov qauv kev nyab xeeb zoo tsim kev nyab xeeb
Pom zoo los ntawm cov koom haum hauv ntiaj teb (piv txwv li, FDA, EMA), nws muaj keeb kwm kev siv tau ntev, nrog kev nkag siab zoo phathokinetics thiab kev ua tau zoo.
Cim npe nrov: Sumatriptan succinate 丨 cas 103628-48-4, Tuam Tshoj sumatriptan succompincinate}}} chaw tsim khoom, cov chaw tsim khoom, Hoobkas

