Olacitinib Malaste 丨 CAS 1208319-27-0

Olacitinib Malaste 丨 CAS 1208319-27-0
Khoom Taw qhia:
Catalog tsis muaj.: Ss124427
CAS TSIS MUAJ .: 1208319-27-0
Purity: 99% min; Assay: 98.0% ~ 102.0%
Khoom npe: Olcacitinib malate
Molecular cov mis: c19h27n5o6s
Molecular hnyav: 453.5
Cov Lus Txhais: N - methyl {{3-dpyrolo2,3-dpyrimidin-4-YL) Aminocyclohexylmethanesulfonamide
Xa kev nug
Kev tsis
Hauj lwm lawm

Hangzhou Leind Chem Co., Ltd. yog ib qho ntawm cov neeg tsim khoom lag luam thiab cov muag khoom ntawm oClacitinib malate 丨 CAS 1208319-27-0 nyob rau hauv Suav teb. Txais tos rau kev lag luam wholesale kev cai ua cov tshuaj lom neeg cov khoom lag luam ntawm cov nqi sib tw los ntawm peb lub hoobkas. Rau cov khoom lag luam pheej yig tshaj, tiv tauj peb tam sim no.

 

Cov lus qhia

 

Kev tshwm sim Tawm - dawb dawb kom dawb hmoov
Kev coj dawb huv 99% min
Lam xav 98.0%~102.0%
Daim qhia npe IR: Qauv Piv Txwv yuav tsum phim cov qauv spectrum
HPLC: Lub sijhawm khaws cia ntawm qhov tseem ceeb tshaj plaws hauv assay npaj sib raug zoo rau cov qauv npaj
So Soluble hauv dmo, insoluble hauv ethyl acetate
Melting taw tes 128 ~ 130 Qib
PH nqi 4.2-5.8
Dej (Kf) 5.0% max
Poob rau ziab 5.0% max
Residue ntawm ignition 0.2% max
Residual cov kuab tshuaj Methanol: 3000 PPM Max
DMF: 860 ppm max
Acetoniturile: 390 ppm max
n - butanol: 3000 ppm max
TetrahyDrofuran: 700 ppm Max
Lwm yam tshuaj Max ib leeg impurity: 0.2% max
Tag nrho cov impurities: 1.0% max

 

 

 

Cov Ntawv Thov

 

OCLacitinib Malaste (CAS 1208319 {4 4}}}}}}}}}} 0) yog ib qho cuam tshuam nrog kev tswj hwm ntawm kev ua xua ntawm dev. Nws ua raws li ib tug xaiv Janus Kinase (JAK) Inhibitor, Modulating lub cev tiv thaiv kab mob tawm thiab kev txo cov mob tshwm sim los ntawm kev ua xua. Olcacitinib Malaste yog cov qauv ntawm qhov ncauj rau cov thawj coj yooj yim xws li cov kab mob entacicitis, thiab lwm yam kev ua xua tsis zoo. Ib qho ntxiv, nws tau siv hauv kev tshawb fawb txog kev kho tsiaj rau kev kawm Jak-stat signaling txoj kev kho mob.

 

Cov txiaj ntsig

 

Cov txiaj ntsig ntawm oClacitinib malate tshwm sim los ntawm nws lub hom phiaj ua haujlwm ntawm kev ua thiab kev pib sai sai ntawm cov nyhuv. Los ntawm xaiv inhibiting inhibiting Jak1 thiab Jak3, nws zoo txo ​​PRO {{ Qhov kev ua si ntawm cov kev ua si ntawm cov kev mob tshwm sim me me piv rau cov corticosteroids lossis lub cev immunosuppressants. Nws muaj cov ncauj lus zoo, tso cai rau cov tsiaj, thiab nws cov kev ua tau zoo thiab kev nyab xeeb profile tau zoo {6} tsim nyob rau hauv kev tshawb nrhiav tsiaj. Nws cov kev xaiv tau tseem ua rau nws muaj txiaj ntsig rau kev tshawb nrhiav rau hauv lub cev tiv thaiv kab mob- Kev kho mob txoj hauv kev.

 

Tag

 

OCLacitinib Malaste yog hom kws kho tsiaj kho mob siv los tswj cov tshuaj tsis haum thiab cov dev. Nws xaiv Jak inhibition muaj kev nyem nrawm los ntawm khaus thiab o thaum txo cov immunosupression. Los ntawm kev sib txuas ua ke, kev nyab xeeb, thiab yooj yim, offine kev xaiv hauv cov tshuaj kho tsiaj thiab cov cuab yeej tshawb fawb hauv kev tshawb fawb muaj txiaj ntsig.

 

 

Cim npe nrov: OCLacitinib Malaste 丨 CASE 1208319-27-0, Tuam Tshoj Oclacitinib Malaste 丨 CAS 1208319-27-0 tuam ntxhab, lwm tus neeg, Hoobkas

Xa kev nug
Tshaj koj qhov kev cia siab
Los ntawm Science mus rau Lub Neej nrog LEAPChem
tiv tauj peb