Cov lus qhia
| Kev tshwm sim | Tawm dawb rau dawb tawv |
| Lam xav | 98% min |
| Ntau tshaj plaws | 0.2% max |
| Tag nrho cov impurities | 1.0% max |
| Poob rau ziab | 1.0% max |
| Residue ntawm ignition | 0.5% max |
Cov Ntawv Thov
Vericiguat (CAS 1350653 {{{-}}}}}}}}}) yog cov tshuaj uas tsis muaj tshuaj Clinically, nws tau thov rau hauv kev kho mob ntawm lub plawv tsis ua haujlwm nrog kev txo cov feem guanosine guanoscet (CGMP) Hauv kev tshawb fawb, Vericiguat tau ua haujlwm los kawm SGC signing pathways mechanisms, thiab kev txhim kho ntawm cov tshiab kev siv tshuaj xyuas cov nitric oxide-cgmp txoj kev. Nws siv txuas ntxiv rau cov kev tshawb fawb ua ntej tshawb xyuas cov kev tiv thaiv ntxas, tiv thaiv cov kev kho mob tiv thaiv kab mob rau lub plawv tsis ua haujlwm.
Cov txiaj ntsig
Cov txiaj ntsig ntawm Vericiguat qia los ntawm nws lub peev xwm los xaiv txhawb kev ua yeeb yam, txhim kho Odogenous Nitric Oxide kev nthuav dav nitric oxide signaling thiab txhawb nqa daim paib end oxostis. Los ntawm kev nce qib CGMP, nws txhim kho lub suab vascular, thiab txhawb cov kev xav tsis zoo rau lub raum tsis ua rau muaj kev nyab xeeb, muab cov ntaub ntawv muaj kev nyab xeeb. Nws qhov rooj ntawm qhov ncauj ntawm qhov ncauj thiab cov khoom siv tshuaj ua ke pub rau cov qauv kev tswj hwm yooj yim thiab kev kho kom zoo sib xws. Vericiguat kuj tseem ua tiav cov kev kho mob plawv uas muaj kev kho mob lub plawv uas muaj kev kho mob, muab cov txiaj ntsig ntxiv rau cov neeg mob uas muaj kev pheej hmoo siab. Nws cov tshuab kev nqis tes ua sawv cev rau txoj kev tsom mus rau lub plawv tsis ua haujlwm ntawm qib molecular signaling, kev txhim kho cov txiaj ntsig kev hloov kho.
Tag
Hauv cov ntsiab lus, Vericiguat yog SGC stimulator siv nyob rau hauv kev kho mob ntawm lub plawv tsis ua hauj lwm thiab kev tshawb fawb plawv. Nws cov ntawv thov suav nrog kev tiv thaiv mob plawv plawv kev tiv thaiv, thiab kev kawm txog kev nyab xeeb ntawm cov txiaj ntsig, thiab kev mob siab rau lwm tus neeg mob siab. Nrog cov yam ntxwv no, Vericiguat yog ib qho kev kho mob tseem ceeb ntawm cov neeg sawv cev thiab tshawb xyuas cov cuab yeej hauv cov hlab ntshav.
Cim npe nrov: Vericiguat 丨 CAS 1350653-205, Tuam Tshoj Vericiguat 丨 CAS 1350653-2053-20-1 Cov Chaw Tsim Tshuaj, Chaw Tsim Tshuaj, Hoobkas

