Hangzhou Leap Chem Co., Ltd. yog ib qho ntawm cov kws tshaj lij thiab cov neeg muag khoom ntawm perindopril arginine 丨cas 612548-45-5 hauv Suav teb. Txais tos rau kev lag luam wholesale kev cai ua cov khoom lag luam ntawm tus nqi sib tw los ntawm peb lub hoobkas. Rau cov khoom pheej yig dua, tiv tauj peb tam sim no.
Specifications
| Qhov tshwm sim | Dawb los yog yuav luag dawb hmoov |
| Kev txheeb xyuas (IR) | Infrared absorption spectrum ntawm cov qauv yuav tsum ua raws li tus qauv |
| Kev txheeb xyuas (HPLC) | Lub sijhawm khaws cia ntawm qhov siab tshaj plaws los ntawm cov qauv kev daws teeb meem sib raug rau qhov kev daws teeb meem, raws li tau txais hauv qhov kev xeem |
| Dej | 5% max |
| Sulfated tshauv | 0.1% max |
| Impurity A (TLC) | 0.25% max |
| Stereochemical purity - Kev tsis haum tshuaj I | 0.1% max |
| Stereochemical purity - Unspecified impurities | 0.1% max |
| Lwm yam tshuaj - Impurity B | 0.3% max |
| Lwm yam tshuaj - Impurity E | 0.4% max |
| Lwm yam tshuaj - Impurity F | 0.2% max |
| Cov tshuaj muaj feem xyuam - Unspecified impurities | 0.1% max |
| Tag nrho impurities | 1% max |
| Cov kuab tshuaj seem - Ethanol | 5000 ppm max |
| Residual kuab tshuaj - Ethyl acetate | 5000 ppm max |
| Cov kuab tshuaj residual - Dichloromethane | 600 ppm max |
| Kev ntsuam xyuas (HPLC) | 98.0% ~ 102.0%. |
Daim ntawv thov
Perindopril arginine yog ib qho tshuaj muaj txiaj ntsig (API) dav siv hauv kev kho mob plawv thiab kev tshawb fawb tshuaj. Nws ua haujlwm raws li angiotensin-hloov enzyme (ACE) inhibitor, pab tswj ntshav siab, plawv tsis ua hauj lwm, thiab txo cov kev pheej hmoo ntawm cov hlab plawv. Hauv kev siv tshuaj kho mob thiab tshuaj, nws tau muab tso rau hauv cov ntsiav tshuaj thiab kev kho mob ua ke kom ntev -lub sij hawm tswj ntshav siab thiab cardioprotection. Hauv kev tsim tshuaj thiab kev tshawb fawb txog kev tsim tshuaj, perindopril arginine yog siv los ua kom zoo dua solubility, bioavailability, thiab stability nyob rau hauv cov ntaub ntawv ntawm qhov ncauj. Nws kuj tseem ua haujlwm raws li cov ntaub ntawv siv hauv kev tshawb fawb pharmacokinetic, kev txhim kho txoj kev tshuaj ntsuam xyuas, thiab kev ntsuas kev tswj xyuas zoo rau ACE inhibitor-raws li kev kho mob.
Cov txiaj ntsig
Cov txiaj ntsig ntawm perindopril arginine tshwm sim los ntawm nws qhov muaj zog ACE inhibition, zoo bioavailability ntawm qhov ncauj, thiab ruaj khov arginine ntsev daim ntawv. Nws txo qis angiotensin II qib, ua rau vasodilation, txhim kho lub plawv, thiab tswj ntshav siab. Cov ntsev arginine txhim kho cov dej solubility thiab tshuaj lom neeg ruaj khov, tso cai rau kev siv tshuaj ntau dua thiab ua kom lub neej ntev ntawm cov tshuaj formulations. Nws cov tshuaj pharmacokinetics uas xav tau kev txhawb nqa ib zaug - kev noj tshuaj txhua hnub, txhim kho kev ua raws li tus neeg mob. Tsis tas li ntawd, perindopril arginine ua kom pom kev sib raug zoo nrog lwm cov tshuaj tiv thaiv kab mob siab, ua kom muaj kev sib xyaw ua ke rau kev tiv thaiv kab mob plawv. Nws qhov zoo-tus yam ntxwv profile ua kom muaj kev tsim tawm thiab kev ntseeg siab hauv kev tshawb fawb thiab kev tsim kho tshuaj.
Xaus
Perindopril arginine yog ib qho tseem ceeb ntawm cov hlab plawv thiab cov tshuaj nruab nrab nrog kev siv hauv kev kho ntshav siab thiab kev kho plawv tsis ua haujlwm. Nws muaj zog ACE inhibition, ruaj khov daim ntawv ntsev, thiab siab bioavailability ua rau nws yog ib qho tseem ceeb compound nyob rau hauv niaj hnub cardiovascular tshuaj. Los ntawm kev txhawb nqa kev tswj ntshav siab, txhim kho kev ua haujlwm ntawm lub plawv, thiab txhim khu kev qha tshuaj, perindopril arginine tseem ua lub luag haujlwm tseem ceeb hauv kev kho mob thiab kev tshawb fawb txog plawv.
Cim npe nrov: perindopril arginine 丨cas 612548-45-5, Tuam Tshoj perindopril arginine丨cas 612548-45-5 manufacturers, lwm tus neeg, Hoobkas

