CAS Nr .: 439239-90-4

CAS Nr .: 439239-90-4
Khoom Taw qhia:
Catalog No.: SS133417 Nr
CAS Nr .: 439239-90-4
Purity: 99% min
Khoom npe: LasMiditan
Cov mis mos molecular: C19H18F3N3O2
Molecular Luj: 377.4
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Kev tsis
Hauj lwm lawm

Hangzhou Leap Chem Co., Ltd. yog ib qho ntawm cov kws tshaj lij thiab cov neeg muag khoom ntawm lasmiditan 丨cas 439239-90-4 hauv Suav teb. Txais tos rau kev lag luam wholesale kev cai ua cov khoom lag luam ntawm tus nqi sib tw los ntawm peb lub hoobkas. Rau cov khoom pheej yig dua, tiv tauj peb tam sim no.

 

Specifications

 

Qhov tshwm sim Yellow rau tawm -dawb hmoov
Purity 99% min
Cov ntsiab lus dej 1% max
Residue ntawm ignition 0.1% max
Cov khoom muaj feem xyuam Ib leeg max tsis paub impurity 0.5% max

 

 

 

Daim ntawv thov

 

Lasmiditan yog ib qho kev xaiv serotonin 5-HT1F receptor agonist siv hauv kev tshawb fawb tshuaj thiab kev siv tshuaj kho mob rau kev kho mob migraine mob. Tsis zoo li cov tshuaj triptans, Lasmiditan tsis ua rau vasoconstriction, ua rau nws tsim nyog rau cov neeg mob uas muaj kev pheej hmoo ntawm cov hlab plawv. Nws yog feem ntau siv rau hauv qhov ncauj formulations kom sai sai ntawm cov tsos mob migraine, nrog rau mob taub hau, xeev siab, thiab rhiab heev rau lub teeb los yog suab. Hauv kev tshawb fawb, Lasmiditan tau ua haujlwm los kawm txog migraine pathophysiology, receptor-specific signaling pathways, thiab kev txhim kho cov tshuaj kho tshiab uas tsom rau cov txheej txheem serotonergic.

 

Cov txiaj ntsig

 

Cov txiaj ntsig ntawm Lasmiditan suav nrog nws qhov kev xaiv siab rau 5-HT1F receptor, uas txo qhov kev pheej hmoo ntawm cov kab mob plawv cuam tshuam nrog cov tshuaj serotonergic tsis xaiv. Nws qhov pib sai sai ua rau muaj txiaj ntsig zoo los ntawm cov tsos mob migraine, txhim kho tus neeg mob lub neej zoo. Qhov sib xyaw ua ke ntawm qhov ncauj bioavailability thiab kev kwv yees cov tshuaj pharmacokinetics ua rau nws yooj yim rau kev siv tshuaj kho mob. Tsis tas li ntawd, Lasmiditan qhov tshwj xeeb receptor tshwj xeeb tso cai rau cov kws tshawb fawb los tshawb nrhiav cov txheej txheem hauv kev kho mob migraine, txhawb kev txhim kho kev nyab xeeb thiab kev kho mob zoo dua rau cov neeg mob sib txawv.

 

Xaus

 

Lasmiditan yog ib qho kev xaiv 5-HT1F receptor agonist siv rau kev kho mob migraine mob thiab kev tshawb fawb tshuaj. Nws qhov tshwj xeeb receptor tshwj xeeb, kev ua tau zoo sai, thiab kev nyab xeeb zoo profile ua rau nws yog ib qho tseem ceeb ntawm kev kho tus neeg sawv cev thiab kev tshawb fawb cov cuab yeej. Cov khoom no txhawb nqa nws lub luag haujlwm hauv kev txhim kho kev tswj hwm migraine thiab nce kev nkag siab ntawm serotonergic signaling nyob rau hauv neurological ntshawv siab.

 

Cim npe nrov: Tuam Tshoj lasmiditan cas 439239-90-4 manufacturers, lwm tus neeg, Hoobkas

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