Oneemilast 丨 CAS 608141-41-9

Oneemilast 丨 CAS 608141-41-9
Khoom Taw qhia:
Catalog tsis muaj .: SS123901
CAS TSIS MUAJ.: 608141-41-9
Purity: 99% min assay: 98% {2}}%
Khoom npe: sanemilast
Molecular cov mis: c22h24n2o7s
Molecular hnyav: 460.5
Txhais tau (s): apemilastum
Xa kev nug
Kev tsis
Hauj lwm lawm

 

Cov lus qhia tshwj xeeb ntawm kev ua haujlwm qub 丨 608141-41-9

 

Kev tshwm sim

Dawb rau lub teeb daj cov crystal

Kev coj dawb huv

99. {0}% min

Lam xav

98% - 102%

Daim qhia npe

IR Pauv thiab Tuav Sij Hawm Ua Haujlwm Nrog Siv

1, {{3- dioxo -2-} isoindolineycetic acid

0. 1% Max

(S) -13-} hydroxy {2}} methyl-methylamide n-acetyl-l-leucine ntsev

0. 1% Max

Tsis paub tus neeg impurity

0. 1% Max

Tag nrho cov impurities

1. {0 max

Melting taw tes

154 - 158 degree

Cov hlau hnyav

10 ppm max

Residue ntawm ignition

0. 1% Max

Acetone

5000 ppm max

Ethanol

5000 ppm max

Dichhloromethane

600 ppm max

Ywg dej

{{0 {}}. 5% Max

Poob rau ziab

{{0 {}}. 5% Max

Chairal Isomers

1. {0 max

 

Cov ntaub ntawv thauj ntawm sendemilast 丨 CAS 608141-41-9

 

Chaw ua uas tsis tau haus

Kev qhia tshwj xeeb

UN NUM

 

Hom

 

Cov Pab Pawg

 

Hs code

2933990099306

Ruaj khov & rov ua

Cov hauv qab no siv rau hauv dav dav los ua cov organic
Cov tshuaj thiab cov khoom sib xyaw sib xyaw: hauv kev sib raug zoo me me, thaum uas tawg ua ib plua plav tawm cov plua plav tawg tuaj yeem xav.

Chaw ntim khoom

Nruj nreem kaw. Qhuav. Combustible cov khoom tau pom zoo cia khoom siv: -25 - -10 degree

Mob kom tsis txhob

 

Lub thawv

 

 

Cov ntaub ntawv kev tsim khoom ntawm apemililast 丨 cas 608141-41-9

 

Chaw ua uas tsis tau haus

Kev qhia tshwj xeeb

Lub peev xwm

 

Hov ntau

 

Lub teb chaws tseem ceeb

 

Peev Xwm \/ Batch

 

Paub lawm

Ntau lawm txij xyoo 2005

Ntxiv rau

Me me rau hauv Tshuag

Praremilast 丨 cas 608141-41-9 yog ib qho orally sortistered me-molecule tshuaj paub rau nws cov tshuaj tiv thaiv kab mob thiab immunomodulatory zog. Nws ua haujlwm raws li xaiv phosphodiesterase 4 (PDE4) Inhibitor thiab feem ntau yog siv nyob rau hauv kev kho mob ntawm autoimmune thiab mob kab mob.

 

Thawj cov ntawv thov ntawm saremilast 丨 cas 608141-41-9

 

1. Psoriasis thiab psoriatic mob caj dab
● Pom zoo kev kho mob rau ib nrab mus rau cov quav hniav loj psorefias.
● Txo cov quav tawv nqaij, ntsuas kev, thiab mob sib koom tes.
● Lwm txoj rau cov kev ua kom raug cai rau cov tshuaj lom neeg; yooj yim txoj cai ntawm qhov ncauj.
2. Beamert tus kab mob
● FDA Pom kev pom zoo rau kev kho mob ntawm qhov ncauj uas cuam tshuam nrog tus kab mob.
● Muaj cov tsos mob zoo tswj tau nrog cov ntaub ntawv kev nyab xeeb nyab xeeb.
3. Thaum igic dermatitis thiab lwm yam teeb meem autoimmune (tshawb xyuas)
● Hauv kev tshawb nrhiav lossis tawm-daim ntawv lo rau:
O atopic dermatitis
o Rheumatoid caj dab
o lupus erythematosus
o mob hnyuv plhaw (IBD)
4. Tej zaum kuj antiviral \/ antifibricotic siv (tawm kev tshawb fawb)
● PDE4 inibitors zoo li sanemililast tau kawm rau lawv lub cev muaj zog-modulating-modulating cov luag haujlwm thiab cov kab mob pulmonary fibrosis).

 

Cov txiaj ntsig ntawm kev kwv yees 丨 cas 608141-41-9

 

✅ daim ntawv ntawm qhov ncauj
Tsis txhob txhaj tshuaj lossis infusions xav tau, txhim kho tus neeg mob kom yooj yim thiab ua raws.
A Hom phiaj immunomodulation
Haign Cytokine signaling tsis muaj kev tiv thaiv kev tiv thaiv kev tiv thaiv kev pheej hmoo, txo qis kev pheej hmoo kis mob thiab mob khees xaws.
✅ Qhov kev zam txim zoo
● Cov kev mob tshwm sim feem ntau muaj mob me rau ntau (piv txwv li, xeev siab, raws plab, mob taub hau) thiab feem ntau daws sijhawm dhau sijhawm.
✅ steroid- thiab biologic-sparing tus neeg sawv cev
● Tso cai txo lossis zam kev corticosteroids thiab txhaj xyoob.

 

Tag

 

Praremilast 丨 cas 608141-41-9 yog ib txoj kev txiav ntawm PDE4 inhiboration qhov ncauj tsis zoo li psoriasis, mob pioriasis, mob pioriatic, thiab coj tus kabmob. Nws qhov kev ua tau zoo, cov ntaub ntawv kev nyab xeeb, thiab txoj haujlwm ntawm qhov ncauj nws yog qhov muaj txiaj ntsig kho tus neeg sawv cev hauv autoimmune thiab mob mob.

 

Cim npe nrov: oneemilast 丨 cas 608141-41-9}}}}}, Tuam Tshoj Sendemilaste 608141-41-9 Cov chaw tsim khoom, cov chaw tsim khoom, Hoobkas

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