Hangzhou Leap Chem Co., Ltd. yog ib qho ntawm cov kws tshaj lij thiab cov neeg muag khoom ntawm thiocolchicoside丨cas 602-41-5 hauv Suav teb. Txais tos rau kev lag luam wholesale kev cai ua cov khoom lag luam ntawm tus nqi sib tw los ntawm peb lub hoobkas. Rau cov khoom pheej yig dua, tiv tauj peb tam sim no.
Specifications
| Kev piav qhia | daj ntseg daj mus rau crystalline hmoov |
| Assay (los ntawm HPLC) | 98.0% -102% (ntawm qhuav hauv paus) |
| Solubility | Soluble hauv dej, me ntsis soluble hauv cawv, insoluble hauv ether thiab acetone |
| Kev txheeb xyuas - IR | IR spectra yuav tsum phim nrog tus qauv |
| Kev txheeb xyuas - UV | Absorbance maxima ntawm 220-440 nm, sib xws nrog tus qauv |
| pH (0.5% w / v sol. hauv dej) | 6.0–7.5 |
| Kev sib hloov kho qhov muag tshwj xeeb (0.5% sol. ntawm 23℃hauv dej) | (-) 550℃rau (-) 580℃(ntawm qhuav hauv paus) |
| Yam Khoom Muaj (los ntawm HPLC) | N-deacetyl N-formyl thiocolchicoside: 0.5% max Colchicoside: 0.5% max Tag nrho tsis paub impurities: 0.5% max |
| Sulfated tshauv | 0.1% max |
| Poob rau ziab | 4.0% max |
| Residual Solvent (Los ntawm GC) | Methanol: 3000 ppm max Ethanol: 5000 ppm max Acetone: 5000 ppm max Chloroform: 60 ppm max |
| Microbial Contamination | 1000 cfu/g max |
| Tag nrho Microbial suav | 100 cfu/g |
| Tag nrho cov poov xab thiab pwm suav | Tsis muaj / g |
| Escherichia coli | Tsis muaj / 10 g |
| Salmonella | Tsis muaj / g |
| Staphylococcus aureus | Tsis muaj / g |
| Cov kab mob endotoxin | 87.5 EU / mg max |
Daim ntawv thov
Thiocolchicoside yog ib nrab -synthetic derivative ntawm colchicoside dav siv nyob rau hauv kws tshuaj rau kev tswj ntawmspasms, spasticity, thiab lwm yam neuromuscular mob. Nws yog feem ntau tsim los rau qhov ncauj, txhaj tshuaj, thiab tshuaj pleev ib ce, muab cov leeg so hauv cov mob xws li mob lumbar, mob ncauj tsev menyuam, thiab tom qab- mob musculoskeletal txhav. Ntxiv rau nws cov kev siv tshuaj kho mob, Thiocolchicoside yog siv hauv kev tshawb fawb tshuaj raws li cov ntaub ntawv siv rau kev kawm neuromuscular kis, receptor binding, thiab cov leeg nqaij relaxant mechanisms. Nws cov qauv tshuaj tso cai rau kev tshawb nrhiav cov qauv-kev sib raug zoo hauv kev txhim kho tom ntej -cov leeg nqaij so thiab cov tshuaj tiv thaiv - cov kab mob.
Cov txiaj ntsig
Cov txiaj ntsig ntawm Thiocolchicoside tshwm sim los ntawm nws cov kev ua haujlwm ntawm cov leeg nqaij muaj zog, kev sib cuam tshuam receptors, thiab cov khoom siv tshuaj muaj txiaj ntsig zoo. Nws ua raws li ib tugGABAergic thiab glycine receptor modulator, muab kev pab zoo ntawm cov leeg nro thiab spasms nrog tsawg kawg hauv nruab nrab paj hlwb sedation piv rau cov leeg nqaij ib txwm so. Nws semi-synthetic xwm ua kom muaj kev ruaj ntseg dua thiab bioavailability piv rau ib txwm tshwm sim colchicoside, tso cai rau cov txiaj ntsig kho tau zoo. Lub compound yog sib xws nrog ntau yam tshuaj formulations, nrog rau cov ntsiav tshuaj, tsiav tshuaj, thiab injectables, enabling yooj nyob rau hauv koob tshuaj thiab kev tswj. Nws qhov zoo -cov tshuaj kho mob tshwj xeeb thiab kev nyab xeeb profile ua rau nws muaj kev ntseeg siab rau ob qho tib si mob thiab mob musculoskeletal mob.
Xaus
Thiocolchicoside yog ib qho tseem ceeb ib nrab- cov leeg nqaij hluavtaws siv dav hauv kev tswj hwm spasticity, musculoskeletal mob, thiab neuromuscular mob. Nws cov kev xaiv receptor kev ua si, tshuaj stability, thiab formulation versatility tso cai rau cov leeg zoo so nrog kev tswj koob tshuaj. Los ntawm kev txhawb nqa kev siv tshuaj kho mob, kev tshawb fawb tshuaj, thiab kev txhim kho cov leeg nqaij zoo dua qub, Thiocolchicoside tseem yog qhov tseem ceeb hauv cov tshuaj niaj hnub thiab kev tshawb fawb tshuaj.
Cim npe nrov: Tuam Tshoj thiocolchicoside cas 602-41-5 manufacturers, lwm tus neeg, Hoobkas

